RT Book, Section A1 Gonzalez, Frank J. A1 Coughtrie, Michael A2 Brunton, Laurence L. A2 Knollmann, Björn C. SR Print(0) ID 1193227030 T1 Drug Metabolism T2 Goodman & Gilman's: The Pharmacological Basis of Therapeutics, 14th Edition YR 2023 FD 2023 PB McGraw-Hill Education PP New York, NY SN 9781264258079 LK hemonc.mhmedical.com/content.aspx?aid=1193227030 RD 2024/03/28 AB AbbreviationsADR: adverse drug reactionAHR: aryl hydrocarbon receptorAUC: area under the plasma concentration–time curveCAR: constitutive androstane receptorCYP: cytochrome P450EH: epoxide hydrolaseER: endoplasmic reticulumFMO: flavin-containing monooxygenaseGI: gastrointestinalGSH and GSSG: reduced and oxidized glutathioneGST: glutathione-S-transferaseHGPRT: hypoxanthine guanine phosphoribosyl transferaseHIF: hypoxia-inducible factorHIV: human immunodeficiency virusINH: isonicotinic acid hydrazide (isoniazid)MAPK: mitogen-activated protein kinasemEH: microsomal epoxide hydrolase6-MP: 6-mercaptopurineMT: methyltransferaseNADPH: nicotinamide adenine dinucleotide phosphateNAPQI:N-acetyl-p-benzoquinone imineNAT:N-acetyltransferasePAPS: 3′-phosphoadenosine-5′-phosphosulfatePPAR: peroxisome proliferator–activated receptorPXR: pregnane X receptorSULT: sulfotransferaseTPMT: thiopurine methyltransferaseUDP-GA: uridine diphosphate–glucuronic acidUGT: uridine diphosphate–glucuronosyltransferase